The Peptide Reference
The Peptide Reference
References
Reference/Tetrapeptide bioregulator

Cortagen

AEDP · Brain Cortex Bioregulator Peptide

research use only

Cortagen is a Khavinson bioregulator tetrapeptide (AEDP) with primary effects on the brain and central nervous system. Developed at Russia's St. Petersburg Institute of Bioregulation and Gerontology, it regulates inflammatory responses in the nervous system, restores balance between pro- and anti-oxidative processes, and stimulates interleukin-2 expression. Research shows potential benefits for ischemic brain injury recovery, nerve regeneration, and reducing autoimmune reactions affecting the CNS.

Regulates central nervous system functionPowerful anti-inflammatory effects in brainSupports nerve regenerationRestores oxidative balance
01

Overview

Cortagen is a Khavinson bioregulator tetrapeptide (AEDP) with primary effects on the brain and central nervous system. Developed at Russia's St. Petersburg Institute of Bioregulation and Gerontology, it regulates inflammatory responses in the nervous system, restores balance between pro- and anti-oxidative processes, and stimulates interleukin-2 expression. Research shows potential benefits for ischemic brain injury recovery, nerve regeneration, and reducing autoimmune reactions affecting the CNS.

Cortagen works through epigenetic regulation by penetrating cell nuclei and interacting with DNA to modulate gene expression. In the heart, it affects genes including Pass1, Hsc70, Bmp2, Wnt4, Eps15, and Eps15-rs. It powerfully regulates inflammatory responses in the nervous system, helping restore proper balance between oxidative and anti-oxidative processes. Cortagen stimulates IL-2 expression and helps regulate immune function, particularly by reducing autoimmune reactions.

02

Research indications

What the compound has been studied for, grouped by body system. Effect size is the reported magnitude where it was measured — not a recommendation.

Neurological Support3
Ischemic Brain Injury Recovery

Shows beneficial long-term results in research following ischemic brain injury.

Moderate
Nerve Regeneration

Research demonstrates effects on restoration of injured nerve function.

Small
Neuroinflammation

Regulates inflammatory response in the nervous system.

Small
Immune Regulation2
Autoimmune Modulation

Helps regulate immune function by reducing autoimmune reactions.

Small
IL-2 Stimulation

Stimulates interleukin-2 expression for immune regulation.

Small
Anti-Aging2
Oxidative Balance

Restores balance between pro- and anti-oxidative processes.

Small
Brain Aging

Addresses age-related CNS changes through bioregulation.

Small
i

A large effect in a weak study and a small effect in a strong one are different things. Effect size is never evidence of use in people.

Quick factsreference only
Class
Tetrapeptide bioregulator
Chain length
4 residues
Molecular weight
416 Da
Typical dose
10-20 mg daily
Frequency
Once daily for 10-20 consecutive days
Cycle length
10-20 days per cycle
Storage
Capsules: room temperature; Injectable lyophilized: 2-8°C; Reconstituted: 2-8°C refrigerated
03

Molecular data

Type
Tetrapeptide bioregulator
Molecular weight
416 Da
Chain length
4 residues
Primary sequenceN → C · 4 residues
H₂N–
AAla1
EGlu2
DAsp3
PPro4
–OH
AEDP
NonpolarPolarAcidicBasic
04

Dosing reference

Doses reported in the literature and by suppliers. These are a record of what has been used in research — reference, never instruction.

ContextRouteAmountFrequency
Standard protocolOral capsules10-20 mgDaily for 10-20 days
MaintenanceOral capsules10 mg2-3 cycles yearly
Research protocolIM or SubQ10 mgDaily for 10 days
05

Interactions

Pinealon

Complementary CNS bioregulators; Cortagen for cortex, Pinealon for general brain.

synergistic
Epitalon

Often combined in comprehensive anti-aging Khavinson protocols.

synergistic
Thymalin

Different organ targets; can be used in comprehensive bioregulator protocols.

compatible
Cardiogen

Part of Khavinson bioregulator family; targets different tissue.

compatible
06

Quality checklist

  • White powder or capsules
  • Clear solution if reconstituted
  • Proper packaging and labeling
  • !Unknown source or purity
  • ×Discoloration
  • ×Unusual odor
  • ×Damaged packaging
07

What to expect

During cycleGene expression modulation begins
Post-cycleEffects persist due to epigenetic changes
Weeks-MonthsNeurological function improvements
Long-termCumulative benefits with periodic cycles
08

Safety

Commonly reported2
  • Generally well-tolerated
  • Minimal side effects reported
Stop and seek advice2
  • Allergic reactions
  • Unusual neurological symptoms
Contraindications3
  • Active neurological emergencies (seek medical care)
  • Known hypersensitivity
  • Pregnancy or breastfeeding
09

FAQ

Is Cortagen helpful for recovery after a stroke or brain injury?

Yes, Cortagen shows research evidence for beneficial effects following ischemic brain injury with long-term improvements in neurological function. It regulates inflammatory responses in nervous tissue and promotes nerve regeneration, making it relevant for post-stroke recovery protocols alongside medical rehabilitation.

How does Cortagen differ from other brain-supporting peptides like Semax?

Cortagen targets the brain cortex specifically through IL-2 stimulation and inflammatory modulation, whereas Semax acts via BDNF upregulation for cognitive effects. Cortagen is more suited for neuroinflammation and recovery, while Semax focuses on cognitive enhancement, and they're often combined in comprehensive protocols.

Can Cortagen help with autoimmune neurological conditions?

Cortagen shows potential for autoimmune modulation through IL-2 regulation and reduction of autoimmune reactions affecting the nervous system. However, the research remains preclinical. Anyone with autoimmune conditions should consult their physician before using, as immune-modulating peptides require careful monitoring.

What's the typical protocol for Cortagen as an anti-aging agent?

Standard anti-aging use involves 10-20mg daily oral capsules for 10-20 consecutive days, repeated 2-3 times yearly. Effects persist post-cycle due to epigenetic changes in gene expression. Some users prefer injectable forms for more direct delivery, though oral bioavailability is generally good for this short peptide.

For research use only. Nothing on this page is medical advice, and no number here is a recommendation to dose.